129. Fangjun Xiong, Haifeng Wang, Lingjie Yan, Lingjun Xu, Yuan Tao, Yan Wu, Fener Chen. Diastereoselective synthesis of pitavastatin calcium via bismuth-catalyzed two-component hemiacetal/oxa-Michael addition reaction. Org. Biomol. Chem., 2015, 13, 9813–9819

128. Haifeng Wang, Linjie Yan, Yan Wu, Yipei Lu, and Fener Chen. Asymmetric Synthesis of Vitamin D3 Analogues: Organocatalytic
Desymmetrization Approach toward the A‑Ring Precursor of Calcifediol. Org. Lett. 2015, 17, 5452−5455

127. Yan Wu, Fang-Jun Xiong, Fen-Er Chen. Stereoselective synthesis of 3-hydroxy-3-methylglutarylecoenzyme A reductase inhibitors. Tetrahedron 2015, 45(71), 8487-8510
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126. Weiqi Chen, Fangjun Xiong, Qian Liu, Lingjun Xu, Yan Wu, Fener Chen. Substrate stereocontrol in bromine-induced intermolecular
cyclization: asymmetric synthesis of pitavastatin calcium. Tetrahedron 2015, 29(71), 4730-4737
.jpg)
125. Chen Zheng, Hai-Feng Wang, Wei-Qi Chen, Wen-Xue Chen, Fen-Er Chen. Organocatalytic Asymmetric Vinylogous Michael Addition of 3-(2-Oxoindolin-3-ylidene)butanoates to Nitroalkenes Catalyzed by a Bifunctional Cinchona-Based Squaramide. Asian J. Org. Chem. 2015, 4(7), 619-621
124. Zheng-Yong Wan, Jin Yao, Tian-Qi Mao, Xin-Long Wang, Hai-Feng Wang,Wen-Xue Chen, Hong Yin, Fen-Er Chen, Erik De Clercq, Dirk Daelemans,Christophe Pannecouque. Pyrimidine sulfonylacetanilides with improved potency against key mutant viruses of HIV-1 by specific targeting of a highly conserved residue. European Journal of Medicinal Chemistry 2015, 12, 215-222

123. Zheng-Yong Wan, Yuan Tao, Ya-Feng Wang, Tian-Qi Mao, Hong Yin, Fen-Er Chen, Hu-Ri Piao, Erik De Clercq, Dirk Daelemans, Christophe Pannecouque. Hybrid chemistry. Part 4: Discovery of etravirine–VRX-480773 hybrids as potent HIV-1 non-nucleoside reverse transcriptase inhibitors. Bioorganic & Medicinal Chemistry 2015, 23, 4248–4255
122. Chen Zheng, Wen-Xue Chen, Fen-Er Chen*, Asymmetric Amination of 3-(2-Oxoindolin-3-ylidene)butanoates Catalyzed by a Cinchona-Derived Alkaloid Asian J. Org. Chem. 2015, 4(10), 1044–1046
121. Tian-Qi Mao, Qiu-Qin He, Zheng-Yong Wan, Wen-Xue Chen, Fen-Er Chen, Gang-Feng Tang, Erik De Clercq c, Dirk Daelemans, Christophe Pannecouque. Anti-HIV diarylpyrimidine–quinolone hybrids and their mode of action. Bioorganic & Medicinal Chemistry 2015, 23, 3860–3868
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120. Hai-Qiu Wu, Jin Yao, Qiu-Qin He, Wen-Xue Chen, Fen-Er Chen, Christophe Pannecouque, Erik De Clercq, Dirk Daelemans. Synthesis and biological evaluation of DAPY–DPEs hybrids as non-nucleoside inhibitors of HIV-1 reverse transcriptase. Bioorg. Med. Chem. 2015(23), 624–631
%20624%E2%80%93631.jpg)
119. Zheng-Yong Wan, Jin Yao, Yuan Tao, Tian-Qi Mao, Xin-Long Wang, Yi-Pei Lu, Hai-Feng Wang, Hong Yin, YanWu, Fen-Er Chen, Erik De Clercq, Dirk Daelemans, Christophe Pannecouque. Discovery of piperidin-4-yl-aminopyrimidine derivatives as potent non-nucleoside HIV-1 reverse transcriptase inhibitors. European Journal of Medicinal Chemistry 2015(97) , 1-9.